Three-component strategy toward 5-membered heterocycles from isocyanide dibromides. LE Kaim, L Grimaud, P Patil Organic letters 13 (5), 1261-1263, 2011 | 80 | 2011 |
Isocyanide 2.0 P Patil, M Ahmadian-Moghaddam, A Dömling Green Chemistry 22 (20), 6902-6911, 2020 | 74 | 2020 |
De novo assembly of highly substituted morpholines and piperazines P Patil, R Madhavachary, K Kurpiewska, J Kalinowska-Tłuścik, ... Organic letters 19 (3), 642-645, 2017 | 45 | 2017 |
Concise Synthesis of Tetrazole–Ketopiperazines by Two Consecutive Ugi Reactions T Zarganes‐Tzitzikas, P Patil, K Khoury, E Herdtweck, A Dömling European journal of organic chemistry 2015 (1), 51-55, 2015 | 40 | 2015 |
Hydrazine in the Ugi tetrazole reaction P Patil, J Zhang, K Kurpiewska, J Kalinowska-Tłuścik, A Dömling Synthesis 48 (08), 1122-1130, 2016 | 37 | 2016 |
MCR synthesis of a tetracyclic tetrazole scaffold P Patil, K Khoury, E Herdtweck, A Dömling Bioorganic & medicinal chemistry 23 (11), 2699-2715, 2015 | 36 | 2015 |
Easy Synthesis of Two Positional Isomeric Tetrazole Libraries Y Wang, P Patil, A Dömling Synthesis 48 (21), 3701-3712, 2016 | 32 | 2016 |
Compounds as dipeptidyl peptidase IV (DPP IV) inhibitors S Arora, N Sinha, P Nair, SK Chakka, A Hajare, A Reddy, P Patil, ... US Patent 8,338,450, 2012 | 30 | 2012 |
Concise synthesis of tetrazole macrocycle EMM Abdelraheem, MP de Haan, P Patil, K Kurpiewska, ... Organic letters 19 (19), 5078-5081, 2017 | 29 | 2017 |
A universal isocyanide for diverse heterocycle syntheses P Patil, K Khoury, E Herdtweck, A Dömling Organic letters 16 (21), 5736-5739, 2014 | 29 | 2014 |
Ugi–Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues L El Kaim, L Grimaud, P Pravin Organic letters 14 (2), 476-478, 2012 | 29 | 2012 |
Combining high‐throughput synthesis and high‐throughput protein crystallography for accelerated hit identification F Sutanto, S Shaabani, R Oerlemans, D Eris, P Patil, M Hadian, M Wang, ... Angewandte Chemie 133 (33), 18379-18387, 2021 | 27 | 2021 |
Diverse Isoquinoline Scaffolds by Ugi/Pomeranz–Fritsch and Ugi/Schlittler–Müller Reactions Y Wang, P Patil, K Kurpiewska, J Kalinowska-Tluscik, A Dömling Organic letters 21 (10), 3533-3537, 2019 | 27 | 2019 |
Multicomponent reaction–derived covalent inhibitor space F Sutanto, S Shaabani, CG Neochoritis, T Zarganes-Tzitzikas, P Patil, ... Science advances 7 (6), eabd9307, 2021 | 26 | 2021 |
Ammonia-promoted one-pot tetrazolopiperidinone synthesis by Ugi reaction P Patil, K Kurpiewska, J Kalinowska-Tłuścik, A Dömling ACS combinatorial science 19 (5), 343-350, 2017 | 25 | 2017 |
Two cycles with one catch: hydrazine in Ugi 4-CR and its postcyclizations Y Wang, P Patil, K Kurpiewska, J Kalinowska-Tluscik, A Dömling ACS Combinatorial Science 19 (3), 193-198, 2017 | 23 | 2017 |
Library-to-library synthesis of highly substituted α-aminomethyl tetrazoles via Ugi reaction P Patil, B Mishra, G Sheombarsing, K Kurpiewska, J Kalinowska-Tłuścik, ... ACS combinatorial science 20 (2), 70-74, 2018 | 20 | 2018 |
Versatile Protecting-Group Free Tetrazolomethane Amine Synthesis by Ugi Reaction P Patil, M de Haan, K Kurpiewska, J Kalinowska-Tłuścik, A Dömling ACS Combinatorial Science 18 (3), 170-175, 2016 | 20 | 2016 |
Sustainability by design: automated nanoscale 2, 3, 4-trisubstituted quinazoline diversity M Hadian, S Shaabani, P Patil, SV Shishkina, H Böltz, A Dömling Green chemistry 22 (8), 2459-2467, 2020 | 19 | 2020 |
Discovery of a highly orally bioavailable c-5-[6-(4-Methanesulfonyloxyphenyl)hexyl]-2-methyl-1,3-dioxane-r-2-carboxylic acid as a potent hypoglycemic and … H Pingali, M Jain, S Shah, S Basu, P Makadia, A Goswami, P Zaware, ... Bioorganic & medicinal chemistry letters 18 (20), 5586-5590, 2008 | 17 | 2008 |