Derek Beauchamp
Derek Beauchamp
Senior Scientist, Janssen R&D
Verified email at
Cited by
Cited by
4-Connected Metal−Organic Assemblies Mediated via Heterochelation and Bridging of Single Metal Ions:  Kagomé Lattice and the M6L12 Octahedron
Y Liu, VC Kravtsov, DA Beauchamp, JF Eubank, M Eddaoudi
Journal of the American Chemical Society 127 (20), 7266-7267, 2005
Hydrogen‐Bonded Networks through Second‐Sphere Coordination
DA Beauchamp, SJ Loeb
Chemistry–A European Journal 8 (22), 5084-5088, 2002
An acetic acid solvate of trimesic acid that exhibits triple inclined interpenetration and mixed supramolecular homosynthons
P Vishweshwar, DA Beauchamp, MJ Zaworotko
Crystal growth & design 6 (11), 2429-2431, 2006
Single-metal-ion-based molecular building blocks (MBBs) approach to the design and synthesis of metal–organic assemblies
JA Brant, Y Liu, DF Sava, D Beauchamp, M Eddaoudi
Journal of molecular structure 796 (1-3), 160-164, 2006
Design and Characterization of Optimized Adenosine A2A/A1 Receptor Antagonists for the Treatment of Parkinson's Disease
BC Shook, S Rassnick, N Wallace, J Crooke, M Ault, D Chakravarty, ...
Journal of medicinal chemistry 55 (3), 1402-1417, 2012
In Vivo Characterization of a Dual Adenosine A2A/A1 Receptor Antagonist in Animal Models of Parkinson’s Disease
BC Shook, S Rassnick, MC Osborne, S Davis, L Westover, J Boulet, ...
Journal of medicinal chemistry 53 (22), 8104-8115, 2010
Molecular squares, rectangles and infinite helical chains utilising the simple ‘corner’ligand 4-(2-pyridyl)-pyrimidine
DA Beauchamp, SJ Loeb
Chemical communications, 2484-2485, 2002
Structure-based design of a benzodiazepine scaffold yields a potent allosteric inhibitor of hepatitis C NS5B RNA polymerase
K Vandyck, MD Cummings, O Nyanguile, CW Boutton, S Vendeville, ...
Journal of medicinal chemistry 52 (14), 4099-4102, 2009
4-Methyl-6,7-dihydro-4H-triazolo[4,5-c]pyridine-Based P2X7 Receptor Antagonists: Optimization of Pharmacokinetic Properties Leading to the Identification of a …
MA Letavic, BM Savall, BD Allison, L Aluisio, JI Andres, M De Angelis, ...
Journal of Medicinal Chemistry 60 (11), 4559-4572, 2017
A novel metal–organic ternary topology constructed from triangular, square and tetrahedral molecular building blocks
GJ McManus, Z Wang, DA Beauchamp, MJ Zaworotko
Chemical communications, 5212-5213, 2007
Benzimidazole modulators of VR1
MR Player, SL Dax, WH Parsons, MR Brandt, RR Calvo, S Patel, J Liu, ...
US Patent 7,951,829, 2011
Aminomethyl substituted thieno [2, 3-d] pyrimidines as adenosine A2A receptor antagonists
BC Shook, D Charavarty, JK Barbay, A Wang, K Leonard, V Alford, ...
MedChemComm 2 (10), 950-965, 2011
Optimization of arylindenopyrimidines as potent adenosine A2A/A1 antagonists
BC Shook, S Rassnick, D Chakravarty, N Wallace, M Ault, J Crooke, ...
Bioorganic & Medicinal Chemistry Letters 20 (9), 2868-2871, 2010
Silver (I) Complexes of 2, 2′; 6′, 4 ″-Terpyridine: The Formation of Discrete Dimers versus Helical Polymers is Anion Dependent
DA Beauchamp, SJ Loeb
Supramolecular Chemistry 17 (8), 617-622, 2005
Indazole-based ligands for estrogen-related receptor α as potential anti-diabetic agents
RJ Patch, H Huang, S Patel, W Cheung, G Xu, BP Zhao, DA Beauchamp, ...
European Journal of Medicinal Chemistry 138, 830-853, 2017
Process development for scale-up of a novel 3, 5-substituted thiazolidine-2, 4-dione compound as a potent inhibitor for estrogen-related receptor 1
X Li, RK Russell, J Spink, S Ballentine, C Teleha, S Branum, K Wells, ...
Organic Process Research & Development 18 (2), 321-330, 2014
Chiral aminocyclopentene-based cycloaddition strategies to bicyclic [3.3. 0] rings
C Cai, FA Kang, DA Beauchamp, Z Sui, RK Russell, CA Teleha
Tetrahedron: Asymmetry 24 (11), 651-656, 2013
An Efficient Synthesis of 3-Substituted N-Glycoside Indoles Useful as Sodium-Dependent Glucose Transporter Inhibitors
X Li, KM Wells, S Branum, S Damon, S Youells, DA Beauchamp, ...
Organic Process Research & Development 16 (11), 1727-1732, 2012
Benzimidazole modulators of vr1
MR Player, SL Dax, WH Parsons, MR Brandt, RR Calvo, S Patel, J Liu, ...
US Patent App. 13/084,718, 2011
Benzimidazole modulators of vr1
MR Player, SL Dax, WH Parsons, MR Brandt, RR Calvo, S Patel, J Liu, ...
US Patent App. 13/084,705, 2011
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