Oxetanes as versatile elements in drug discovery and synthesis JA Burkhard, G Wuitschik, M Rogers‐Evans, K Müller, EM Carreira Angewandte Chemie International Edition 49 (48), 9052-9067, 2010 | 412 | 2010 |
Oxetanes in drug discovery: structural and synthetic insights G Wuitschik, EM Carreira, B Wagner, H Fischer, I Parrilla, F Schuler, ... Journal of medicinal chemistry 53 (8), 3227-3246, 2010 | 384 | 2010 |
Oxetanes as promising modules in drug discovery G Wuitschik, M Rogers‐Evans, K Müller, H Fischer, B Wagner, F Schuler, ... Angewandte Chemie International Edition 45 (46), 7736-7739, 2006 | 258 | 2006 |
Spirocyclic oxetanes: synthesis and properties G Wuitschik, M Rogers-Evans, A Buckl, M Bernasconi, M Marki, T Godel, ... Angewandte Chemie 120 (24), 4588, 2008 | 220 | 2008 |
Piperazic acid-containing natural products: isolation, biological relevance and total synthesis AJ Oelke, DJ France, T Hofmann, G Wuitschik, SV Ley Natural Product Reports 28 (8), 1445-1471, 2011 | 90 | 2011 |
Synthesis and stability of oxetane analogs of thalidomide and lenalidomide JA Burkhard, G Wuitschik, JM Plancher, M Rogers-Evans, EM Carreira Organic letters 15 (17), 4312-4315, 2013 | 87 | 2013 |
Oxetane als vielseitige Bausteine in der Wirkstoff‐Forschung und Synthese JA Burkhard, G Wuitschik, M Rogers‐Evans, K Müller, EM Carreira Angewandte Chemie 122 (48), 9236-9251, 2010 | 85 | 2010 |
A Ru-Catalyzed Tandem Alkyne−Enone Coupling/Michael Addition: Synthesis of 4-Methylene-2,6-cis-tetrahydropyrans BM Trost, H Yang, G Wuitschik Organic Letters 7 (21), 4761-4764, 2005 | 70 | 2005 |
Total synthesis of chloptosin AJ Oelke, DJ France, T Hofmann, G Wuitschik, SV Ley Angewandte Chemie International Edition 49 (35), 6139-6142, 2010 | 57 | 2010 |
Total synthesis of chloptosin: A dimeric cyclohexapeptide AJ Oelke, F Antonietti, L Bertone, PB Cranwell, DJ France, RJM Goss, ... Chemistry–A European Journal 17 (15), 4183-4194, 2011 | 51 | 2011 |
What can reaction databases teach us about Buchwald–Hartwig cross-couplings? M Fitzner, G Wuitschik, RJ Koller, JM Adam, T Schindler, JL Reymond Chemical science 11 (48), 13085-13093, 2020 | 46 | 2020 |
A Robust, Recyclable Resin for Decagram Scale Resolution of (±)‐Mefloquine and Other Chiral N‐Heterocycles I Kreituss, KY Chen, SH Eitel, JM Adam, G Wuitschik, A Fettes, JW Bode Angewandte Chemie International Edition 55 (4), 1553-1556, 2016 | 24 | 2016 |
Using data analysis to evaluate and compare chemical syntheses D Kaiser, J Yang, G Wuitschik Organic Process Research & Development 22 (9), 1222-1235, 2018 | 23 | 2018 |
The search for tricyanomethane (cyanoform) D Šišak, LB McCusker, A Buckl, G Wuitschik, YL Wu, WB Schweizer, ... Chemistry–A European Journal 16 (24), 7224-7230, 2010 | 22 | 2010 |
Enabling late-stage drug diversification by high-throughput experimentation with geometric deep learning DF Nippa, K Atz, R Hohler, AT Müller, A Marx, C Bartelmus, G Wuitschik, ... Nature Chemistry 16 (2), 239-248, 2024 | 17 | 2024 |
Machine Learning C–N Couplings: Obstacles for a General-Purpose Reaction Yield Prediction M Fitzner, G Wuitschik, R Koller, JM Adam, T Schindler ACS omega 8 (3), 3017-3025, 2023 | 16 | 2023 |
Oxetanes in drug discovery G Wuitschik ETH Zurich, 2008 | 15 | 2008 |
Tricyanomethane and its salts with nitrogen bases: A correction of sixteen reports K Banert, M Hagedorn Synlett 30 (12), 1427-1430, 2019 | 14 | 2019 |
Accounting for different reactivities of sulfinate and thiosulfate salts in regioselective azetidine coupling via C–H sulfenylation of indoles MAE Al-Saedy, ACMA Nassoy, JPA Harrity Synlett 29 (03), 349-353, 2018 | 7 | 2018 |
Oxetan‐3‐one: Chemistry and Synthesis G Wuitschik, EM Carreira, M Rogers‐Evans, K Muller ChemInform 40 (13), no-no, 2009 | 7 | 2009 |