Recent progress in diaryl ether synthesis D Kikelj Synthesis 2006 (14), 2271-2285, 2006 | 187 | 2006 |
Recent advances in the synthesis of 2H-1, 4-benzoxazin-3-(4H)-ones and 3, 4-dihydro-2H-1, 4-benzoxazines J Ilaš, PŠ Anderluh, MS Dolenc, D Kikelj Tetrahedron 61 (31), 7325-7348, 2005 | 186 | 2005 |
Dual inhibitors of human DNA topoisomerase II and other cancer-related targets Z Skok, N Zidar, D Kikelj, J Ilaš Journal of medicinal chemistry 63 (3), 884-904, 2019 | 163 | 2019 |
Efflux pump inhibitors of clinically relevant multidrug resistant bacteria A Lamut, L Peterlin Mašič, D Kikelj, T Tomašič Medicinal Research Reviews 39 (6), 2460-2504, 2019 | 157 | 2019 |
Arginine mimetics L Peterlin-Mašič, D Kikelj Tetrahedron 57 (33), 7073-7105, 2001 | 144 | 2001 |
Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site T Tomasic, S Katsamakas, Z Hodnik, J Ilaš, M Brvar, T Solmajer, ... Journal of medicinal chemistry 58 (14), 5501-5521, 2015 | 124 | 2015 |
Discovery of benzothiazole scaffold-based DNA gyrase B inhibitors M Gjorgjieva, T Tomasic, M Barancokova, S Katsamakas, J Ilas, ... Journal of medicinal chemistry 59 (19), 8941-8954, 2016 | 123 | 2016 |
Discovery of novel 5-benzylidenerhodanine and 5-benzylidenethiazolidine-2, 4-dione inhibitors of MurD ligase N Zidar, T Tomašić, R Šink, V Rupnik, A Kovac, S Turk, D Patin, ... Journal of medicinal chemistry 53 (18), 6584-6594, 2010 | 121 | 2010 |
5‐Benzylidenethiazolidin‐4‐ones as multitarget inhibitors of bacterial Mur ligases T Tomašić, N Zidar, A Kovač, S Turk, M Simčič, D Blanot, ... ChemMedChem: Chemistry Enabling Drug Discovery 5 (2), 286-295, 2010 | 94 | 2010 |
Synthesis and antibacterial activity of 5-ylidenethiazolidin-4-ones and 5-benzylidene-4, 6-pyrimidinediones T Tomašić, N Zidar, M Mueller-Premru, D Kikelj, LP Mašič European Journal of Medicinal Chemistry 45 (4), 1667-1672, 2010 | 85 | 2010 |
Toward a Novel Class of Antithrombotic Compounds with Dual Function. Discovery of 1,4-Benzoxazin-3(4H)-one Derivatives Possessing Thrombin Inhibitory and … P Štefanič Anderluh, M Anderluh, J Ilaš, J Mravljak, M Sollner Dolenc, ... Journal of medicinal chemistry 48 (9), 3110-3113, 2005 | 77 | 2005 |
Antimicrobial activity of the marine alkaloids, clathrodin and oroidin, and their synthetic analogues N Zidar, S Montalvão, Ž Hodnik, DA Nawrot, A Žula, J Ilaš, D Kikelj, ... Marine drugs 12 (2), 940-963, 2014 | 70 | 2014 |
3,4-Dihydro-2H-1,4-benzoxazine Derivatives Combining Thrombin Inhibitory and Glycoprotein IIb/IIIa Receptor Antagonistic Activity as a Novel Class of … J Ilaš, Z Jakopin, T Borštnar, M Stegnar, D Kikelj Journal of medicinal chemistry 51 (18), 5617-5629, 2008 | 69 | 2008 |
Phosphonate inhibitors of antigen 85C, a crucial enzyme involved in the biosynthesis of the Mycobacterium tuberculosis cell wall S Gobec, I Plantan, J Mravljak, RA Wilson, GS Besra, D Kikelj Bioorganic & medicinal chemistry letters 14 (13), 3559-3562, 2004 | 68 | 2004 |
N-Phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and Evaluation N Zidar, H Macut, T Tomasic, M Brvar, S Montalvao, P Tammela, ... Journal of medicinal chemistry 58 (15), 6179-6194, 2015 | 64 | 2015 |
Synthesis and biological evaluation of new glutamic acid-based inhibitors of MurD ligase T Tomašić, N Zidar, V Rupnik, A Kovač, D Blanot, S Gobec, D Kikelj, ... Bioorganic & Medicinal Chemistry Letters 19 (1), 153-157, 2009 | 63 | 2009 |
Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors Ž Jakopin, J Ilaš, M Barančoková, M Brvar, P Tammela, MS Dolenc, ... European Journal of Medicinal Chemistry 130, 171-184, 2017 | 62 | 2017 |
Structure-Based Design of a New Series of d-Glutamic Acid Based Inhibitors of Bacterial UDP-N-acetylmuramoyl-l-alanine:d-glutamate Ligase (MurD) T Tomašić, N Zidar, R Sink, A Kovač, D Blanot, C Contreras-Martel, ... Journal of medicinal chemistry 54 (13), 4600-4610, 2011 | 62 | 2011 |
The application of Freidinger lactams and their analogs in the design of conformationally constrained peptidomimetics A Perdih, D Kikelj Current medicinal chemistry 13 (13), 1525-1556, 2006 | 61 | 2006 |
Design, synthesis, biochemical evaluation and antimycobacterial action of phosphonate inhibitors of antigen 85C, a crucial enzyme involved in biosynthesis of the mycobacterial … S Gobec, I Plantan, J Mravljak, U Švajger, RA Wilson, GS Besra, ... European journal of medicinal chemistry 42 (1), 54-63, 2007 | 60 | 2007 |