| The reluctant polymorph: investigation into the effect of self-association on the solvent mediated phase transformation and nucleation of theophylline R Bobrovs, L Seton, N Dempster CrystEngComm 17 (28), 5237-5251, 2015 | 50 | 2015 |
| Potent SARS-CoV-2 mRNA cap methyltransferase inhibitors by bioisosteric replacement of methionine in SAM cosubstrate O Bobileva, R Bobrovs, I Kanepe, L Patetko, G Kalnins, M Sisovs, AL Bula, ... ACS Medicinal Chemistry Letters 12 (7), 1102-1107, 2021 | 40 | 2021 |
| Targeting bacterial Sortase A with covalent inhibitors: 27 new starting points for structure-based hit-to-lead optimization K Jaudzems, V Kurbatska, A Je̅kabsons, R Bobrovs, Z Rudevica, ... ACS Infectious Diseases 6 (2), 186-194, 2019 | 25 | 2019 |
| Peptidomimetic plasmepsin inhibitors with potent anti-malarial activity and selectivity against cathepsin D R Zogota, L Kinena, C Withers-Martinez, MJ Blackman, R Bobrovs, ... European Journal of Medicinal Chemistry 163, 344-352, 2019 | 25 | 2019 |
| Solvent-mediated phase transformation between two tegafur polymorphs in several solvents R Bobrovs, L Seton, A Actiņš CrystEngComm 16 (46), 10581-10591, 2014 | 24 | 2014 |
| Discovery of SARS-CoV-2 Nsp14 and Nsp16 methyltransferase inhibitors by high-throughput virtual screening R Bobrovs, I Kanepe, N Narvaiss, L Patetko, G Kalnins, M Sisovs, AL Bula, ... Pharmaceuticals 14 (12), 1243, 2021 | 22 | 2021 |
| Polymorph-Selective Role of Hydrogen Bonding and π–π Stacking in p-Aminobenzoic Acid Solutions R Bobrovs, L Drunka, AA Auzins, K Jaudzems, M Salvalaglio Crystal Growth & Design 21 (1), 436-448, 2020 | 22 | 2020 |
| Exploiting structural dynamics to design open-flap inhibitors of malarial aspartic proteases R Bobrovs, K Jaudzems, A Jirgensons Journal of Medicinal Chemistry 62 (20), 8931-8950, 2019 | 21 | 2019 |
| Formation and transformations of organic salt hydrates: Four encenicline hydrochloride monohydrates and respective isostructural desolvates R Bobrovs, A Kons, A Berzins, T Rekis, A Actins Crystal Growth & Design 18 (4), 2100-2111, 2018 | 14 | 2018 |
| 2-Aminoquinazolin-4 (3H)-one based plasmepsin inhibitors with improved hydrophilicity and selectivity D Rasina, G Stakanovs, OV Borysov, T Pantelejevs, R Bobrovs, ... Bioorganic & Medicinal Chemistry 26 (9), 2488-2500, 2018 | 12 | 2018 |
| Ultrafast Fragment Screening Using Photo-Hyperpolarized (CIDNP) NMR F Torres, M Bütikofer, GR Stadler, A Renn, H Kadavath, R Bobrovs, ... Journal of the American Chemical Society 145 (22), 12066-12080, 2023 | 10 | 2023 |
| Azole‐based non‐peptidomimetic plasmepsin inhibitors L Kinena, G Leitis, I Kanepe‐Lapsa, R Bobrovs, K Jaudzems, V Ozola, ... Archiv der Pharmazie 351 (9), 1800151, 2018 | 10 | 2018 |
| 3-(Adenosylthio) benzoic acid derivatives as SARS-CoV-2 Nsp14 methyltransferase inhibitors O Bobileva, R Bobrovs, EE Sirma, I Kanepe, AL Bula, L Patetko, ... Molecules 28 (2), 768, 2023 | 8 | 2023 |
| trans-Fluorine Effect in Cyclopropane: Diastereoselective Synthesis of Fluorocyclopropyl Cabozantinib Analogs J Veliks, M Videja, A Kinens, R Bobrovs, M Priede, J Kuka ACS Medicinal Chemistry Letters 11 (11), 2146-2150, 2020 | 8 | 2020 |
| Three anhydrous forms and a dihydrate form of quifenadine hydrochloride: a structural study of the thermodynamic stability and dehydration mechanism A Kons, L Rutkovska, A Bērziņš, R Bobrovs, A Actiņš CrystEngComm 17 (19), 3627-3635, 2015 | 8 | 2015 |
| Organic solvents vapor pressure and relative humidity effects on the phase transition rate of α and β forms of tegafur S Petkune, R Bobrovs, A Actiņ š Pharmaceutical Development and Technology 17 (5), 625-631, 2012 | 7 | 2012 |
| Aggregation Condition–Structure Relationship of Mouse Prion Protein Fibrils J Fridmanis, Z Toleikis, T Sneideris, M Ziaunys, R Bobrovs, V Smirnovas, ... International journal of molecular sciences 22 (17), 9635, 2021 | 5 | 2021 |
| Synthesis of 2-aminopyridopyrimidinones and their plasmepsin I, II, IV inhibition potency D Rasina, G Stakanovs, I Kanepe-Lapsa, R Bobrovs, K Jaudzems, ... Chemistry of Heterocyclic Compounds 56, 786-792, 2020 | 5 | 2020 |
| Optimization of sample preparation conditions for detecting trace amounts of β‐tegafur in α‐and β‐tegafur mixture R Bobrovs, A Actiņš Journal of Pharmaceutical Sciences, 2012 | 5 | 2012 |
| Exploring aspartic protease inhibitor binding to design selective antimalarials R Bobrovs, EE Basens, L Drunka, I Kanepe, S Matisone, KK Velins, ... Journal of Chemical Information and Modeling 62 (13), 3263-3273, 2022 | 4 | 2022 |
Agris BērziņšUniversity of LatviaGeverifieerd e-mailadres voor lu.lv
