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Stamatia Vassiliou
Stamatia Vassiliou
National and Kapodistrian University of Athens, Department of Chemistry, Laboratory of Organic
Verified email at chem.uoa.gr
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Cited by
Year
RXP 407, a phosphinic peptide, is a potent inhibitor of angiotensin I converting enzyme able to differentiate between its two active sites
V Dive, J Cotton, A Yiotakis, A Michaud, S Vassiliou, J Jiracek, G Vazeux, ...
Proceedings of the National Academy of Sciences 96 (8), 4330-4335, 1999
2161999
Structure of astacin with a transition-state analogue inhibitor
F Grams, V Dive, A Yiotakis, I Yiallouros, S Vassiliou, R Zwilling, W Bode, ...
Nature structural biology 3 (8), 671-675, 1996
1981996
Phosphinic pseudo-tripeptides as potent inhibitors of matrix metalloproteinases: a structure− activity study
S Vassiliou, A Mucha, P Cuniasse, D Georgiadis, K Lucet-Levannier, ...
Journal of medicinal chemistry 42 (14), 2610-2620, 1999
1411999
RXP 407, a selective inhibitor of the N-domain of angiotensin I-converting enzyme, blocks in vivo the degradation of hemoregulatory peptide acetyl-Ser-Asp-Lys-Pro with no …
C Junot, MF Gonzales, E Ezan, J Cotton, G Vazeux, A Michaud, M Azizi, ...
Journal of pharmacology and experimental therapeutics 297 (2), 606-611, 2001
1382001
Design, synthesis, and evaluation of novel organophosphorus inhibitors of bacterial ureases
S Vassiliou, A Grabowiecka, P Kosikowska, A Yiotakis, P Kafarski, ...
Journal of Medicinal Chemistry 51 (18), 5736-5744, 2008
1062008
Protection of the hydroxyphosphinyl function of phosphinic dipeptides by adamantyl. Application to the solid-phase synthesis of phosphinic peptides
A Yiotakis, S Vassiliou, J Jiráček, V Dive
The Journal of organic chemistry 61 (19), 6601-6605, 1996
961996
An effective one-pot synthesis of 3-benzylfurans and their potential utility as versatile precursors of 3, 4-dibenzyltetrahydrofuran lignans. Formal synthesis of (±)-burseran
S Garçon, S Vassiliou, M Cavicchioli, B Hartmann, N Monteiro, G Balme
The Journal of Organic Chemistry 66 (11), 4069-4073, 2001
712001
Computer-aided optimization of phosphinic inhibitors of bacterial ureases
S Vassiliou, P Kosikowska, A Grabowiecka, A Yiotakis, P Kafarski, ...
Journal of medicinal chemistry 53 (15), 5597-5606, 2010
652010
The M18 aspartyl aminopeptidase of the human malaria parasite Plasmodium falciparum
F Teuscher, J Lowther, TS Skinner-Adams, T Spielmann, MWA Dixon, ...
Journal of Biological Chemistry 282 (42), 30817-30826, 2007
652007
Phosphinic peptides, the first potent inhibitors of astacin, behave as extremely slow-binding inhibitors
I Yiallouros, S Vassiliou, A Yiotakis, R Zwilling, W Stöcker, V Dive
Biochemical Journal 331 (2), 375-379, 1998
631998
Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases
S Vassiliou, E Weglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, ...
Journal of medicinal chemistry 57 (19), 8140-8151, 2014
602014
A convenient method to synthesize phosphinic peptides containing an aspartyl or glutamyl aminophosphinic acid. Use of the phenyl group as the carboxyl synthon
D Georgiadis, M Matziari, S Vassiliou, V Dive, A Yiotakis
Tetrahedron 55 (51), 14635-14648, 1999
591999
A synthetic method for diversification of the P1′ substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1′ binding pockets of leucine …
S Vassiliou, M Xeilari, A Yiotakis, J Grembecka, M Pawełczak, P Kafarski, ...
Bioorganic & medicinal chemistry 15 (9), 3187-3200, 2007
442007
Phosphinic peptide inhibitors as tools in the study of the function of zinc metallopeptidases.
V Dive, K Lucet-Levannier, D Georgiadis, J Cotton, S Vassiliou, ...
Biochemical Society Transactions 28 (4), 455-460, 2000
392000
Cyclic peptides with a phosphinic bond as potent inhibitors of a zinc bacterial collagenase
A Yiotakis, A Lecoq, S Vassiliou, I Raynal, P Cuniasse, V Dive
Journal of medicinal chemistry 37 (17), 2713-2720, 1994
381994
Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues
E Węglarz-Tomczak, S Vassiliou, A Mucha
Bioorganic & Medicinal Chemistry Letters 26 (16), 4122-4126, 2016
312016
Integrated Transition Metal Catalysed Reactions: Synthesis of Polysubstituted 4‐(Phenoxymethyl)‐3‐pyrrolines and Their Isomers by One‐Pot Coupling of Propargylamines, Vinyl …
B Clique, S Vassiliou, N Monteiro, G Balme
European Journal of Organic Chemistry 2002 (9), 1493-1499, 2002
292002
Novel anti-Alzheimer phenol-lipoyl hybrids: Synthesis, physico-chemical characterization, and biological evaluation
A Pagoni, L Marinelli, A Di Stefano, M Ciulla, H Turkez, A Mardinoglu, ...
European Journal of Medicinal Chemistry 186, 111880, 2020
212020
Covalent inhibition of bacterial urease by bifunctional catechol-based phosphonates and phosphinates
A Pagoni, A Grabowiecka, W Tabor, A Mucha, S Vassiliou, Ł Berlicki
Journal of Medicinal Chemistry 64 (1), 404-416, 2020
202020
Three component Kabachnik-Fields condensation leading to substituted aminomethane-P-hydroxymethylphosphonic acids as a tool for screening of bacterial urease inhibitors
S Vassiliou, A Grabowiecka, P Kosikowska, Ł Berlicki
Arkivoc 4, 33-43, 2012
202012
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