A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than Δ9-tetrahydrocannabinol: Δ9-Tetrahydrocannabiphorol C Citti, P Linciano, F Russo, L Luongo, M Iannotta, S Maione, A Laganà, ... Scientific reports 9 (1), 1-13, 2019 | 180 | 2019 |
Ten years with New Delhi metallo-β-lactamase-1 (NDM-1): from structural insights to inhibitor design P Linciano, L Cendron, E Gianquinto, F Spyrakis, D Tondi ACS infectious diseases 5 (1), 9-34, 2018 | 138 | 2018 |
Cannabinoid profiling of hemp seed oil by liquid chromatography coupled to high-resolution mass spectrometry C Citti, P Linciano, S Panseri, F Vezzalini, F Forni, MA Vandelli, ... Frontiers in Plant Science 10, 120, 2019 | 125 | 2019 |
Analysis of impurities of cannabidiol from hemp. Isolation, characterization and synthesis of cannabidibutol, the novel cannabidiol butyl analog C Citti, P Linciano, F Forni, MA Vandelli, G Gigli, A Laganà, G Cannazza Journal of Pharmaceutical and Biomedical Analysis 175, 112752, 2019 | 67 | 2019 |
Isolation of a high-affinity cannabinoid for the human CB1 receptor from a medicinal Cannabis sativa variety: Δ9-tetrahydrocannabutol, the butyl homologue of Δ9 … P Linciano, C Citti, L Luongo, C Belardo, S Maione, MA Vandelli, F Forni, ... Journal of natural products 83 (1), 88-98, 2019 | 58 | 2019 |
Identification of a new cannabidiol n-hexyl homolog in a medicinal cannabis variety with an antinociceptive activity in mice: Cannabidihexol P Linciano, C Citti, F Russo, F Tolomeo, A Laganà, AL Capriotti, L Luongo, ... Scientific Reports 10 (1), 22019, 2020 | 42 | 2020 |
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections P Linciano, CB Moraes, LM Alcantara, CH Franco, B Pascoalino, ... European Journal of Medicinal Chemistry 146, 423-434, 2018 | 37 | 2018 |
Structural development studies of PPARs ligands based on tyrosine scaffold B De Filippis, P Linciano, A Ammazzalorso, C Di Giovanni, M Fantacuzzi, ... European Journal of Medicinal Chemistry 89, 817-825, 2015 | 36 | 2015 |
Synthesis and structure–activity relationships of fibrate-based analogues inside PPARs L Giampietro, A D’Angelo, A Giancristofaro, A Ammazzalorso, ... Bioorganic & medicinal chemistry letters 22 (24), 7662-7666, 2012 | 35 | 2012 |
Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To Inhibit Trypanosoma brucei Pteridine Reductase in Support of Early-Stage Drug Discovery P Linciano, A Dawson, I Pöhner, DM Costa, MS Sa, A Cordeiro-da-Silva, ... ACS omega 2 (9), 5666-5683, 2017 | 30 | 2017 |
Enhancement of benzothiazoles as pteridine reductase-1 inhibitors for the treatment of trypanosomatidic infections P Linciano, C Pozzi, LD Iacono, F di Pisa, G Landi, A Bonucci, S Gul, ... Journal of Medicinal Chemistry 62 (8), 3989-4012, 2019 | 27 | 2019 |
Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC‐2: A Step against Bacterial Resistance G Celenza, M Vicario, P Bellio, P Linciano, M Perilli, A Oliver, J Blazquez, ... ChemMedChem 13 (7), 713-724, 2018 | 27 | 2018 |
Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds C Borsari, N Santarem, J Torrado, AI Olías, MJ Corral, C Baptista, S Gul, ... European Journal of Medicinal Chemistry 126, 1129-1135, 2017 | 26 | 2017 |
Origin of Δ9-Tetrahydrocannabinol Impurity in Synthetic Cannabidiol C Citti, F Russo, P Linciano, SS Strallhofer, F Tolomeo, F Forni, ... Cannabis and cannabinoid research 6 (1), 28-39, 2021 | 22 | 2021 |
Tackling antimicrobial resistance with small molecules targeting LsrK: Challenges and opportunities P Linciano, V Cavalloro, E Martino, J Kirchmair, R Listro, D Rossi, ... Journal of Medicinal Chemistry 63 (24), 15243-15257, 2020 | 22 | 2020 |
Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and … C Borsari, MD Jiménez-Antón, J Eick, E Bifeld, JJ Torrado, ... European Journal of Medicinal Chemistry 183, 111676, 2019 | 22 | 2019 |
Accelerating drug discovery efforts for trypanosomatidic infections using an integrated transnational academic drug discovery platform CB Moraes, G Witt, M Kuzikov, B Ellinger, T Calogeropoulou, KC Prousis, ... SLAS DISCOVERY: Advancing Life Sciences R&D 24 (3), 346-361, 2019 | 22 | 2019 |
Fibrate-derived N-(methylsulfonyl) amides with antagonistic properties on PPARα A Ammazzalorso, A D'Angelo, A Giancristofaro, B De Filippis, M Di Matteo, ... European journal of medicinal chemistry 58, 317-322, 2012 | 22 | 2012 |
1, 3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity S Franchini, C Sorbi, P Linciano, G Carnevale, A Tait, S Ronsisvalle, ... European Journal of Medicinal Chemistry 176, 310-325, 2019 | 20 | 2019 |
Use of Primary Amines for the Selective N-Alkylation of Anilines by a Reusable Heterogeneous Catalyst P Linciano, M Pizzetti, A Porcheddu, M Taddei Synlett 24 (17), 2249-2254, 2013 | 20 | 2013 |